Citation: Jian Ping LI, Qian Fu LUO, Yu Min SONG, Yu Lu WANG. A Rapid and Efficient Synthesis of Diaryl Thioureas via Solvent-Free Reaction Using Microwave[J]. Chinese Chemical Letters, ;2001, 12(5): 383-386. shu

A Rapid and Efficient Synthesis of Diaryl Thioureas via Solvent-Free Reaction Using Microwave

College of Chemistry & Environmental Science, Henan Normal University, Xinxiang 453002 Key Laboratory of Environmental Science & Engineering of Henan Education Commission, Xinxiang 453002

Received Date: 8 October 2000

Fund Project: We are grateful for the financial support from the Key Laboratory of Environmental Science and Engineering of Henan Education Commission.

A rapid and efficient method for the preparation of diaryl thiourea compounds was reported for the first time.Twelve diaryl thiourea compounds that possessing biological activity have been synthesized in excellent yields (91-97%).The reaction proved to be extremely simple and highly efficient (in 1.5-4.5 min).
- Diaryl thiourea,
- microwave technique,
- solvent-free reaction.
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